In vitro screening of UGT2B10 in silico prioritized putative ligands from drugs used in the pediatric hematopoietic stem cell transplantation setting

Screening in vitro of acetaminophen, lorazepam, mycophenolic acid and voriconazole N-oxide to assess the potential of being substrates and/or inhibitors of UGT2B10

Organizational unit: Laboratoire de Pharmacologie et Toxicologie cliniques

Type: Dataset

DOI: 10.26037/yareta:4f2kuon35jc27opnijubgqkmge

License: Creative Commons Attribution 4.0 International

Keywords: In vitro, UHPLC, UGT, MS

Publication date

04/09/2024

Retention date02/09/2034

Access levelPublic

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Contributors

Bennani, Yahia

Ben Hassine, Khalil

Gencaslan, Muhammed

Boudal-Khosbheen, Mary

Samer, Caroline

Ansari, Marc

Daali, Youssef

Uppugunduri Satyanarayana, Chakradhara Rao

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Metadata version: 3.1

Disposal approval: Yes

Retention expiration: 02/09/2034 00:00:00

Created: 04/09/2024 10:06:30

Deposit: In vitro screening of UGT2B10 in silico prioritized putative ligands from drugs used in the pediatric hematopoietic stem cell transplantation setting

Deposit creation

Deposit approval: 04/09/2024 10:06:26

SIP: In vitro screening of UGT2B10 in silico prioritized putative ligands from drugs used in the pediatric hematopoietic stem cell transplantation setting

AIP: In vitro screening of UGT2B10 in silico prioritized putative ligands from drugs used in the pediatric hematopoietic stem cell transplantation setting

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In vitro screening of UGT2B10 in silico prioritized putative ligands from drugs used in the pediatric hematopoietic stem cell transplantation setting

Screening in vitro of acetaminophen, lorazepam, mycophenolic acid and voriconazole N-oxide to assess the potential of being substrates and/or inhibitors of UGT2B10

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